TIK-301
MedChemExpress
Description: TIK-301 (PD-6735) is a chlorinated melatonin derivative and a potent, high-affinity and orally active melatonin MT1 and MT2 receptors agonist with Kis of 0.081 nM and 0.042 nM, respectively. TIK-301 is also a 5-HT2B/5-HT2C receptors antagonist with antidepressant action. TIK-301 has the potential for sleep disorders and other circadian rhythm disorders treatment[1][2][3].
CAS number: 118702-11-7
Formula: C14H17ClN2O2
Solubility: 10 mM in DMSO
SMILES: CC(NC[C@@H](C1=CNC2=C1C=C(OC)C(Cl)=C2)C)=O
Molecular Weight: 280.75
Applications: Neuroscience-Neuromodulation
For research use only. Not to be used for human or animal treatment or consumption.